SCHEMBL13622865

SCHEMBL13622865

CN1CC(N2CCc3cc(-n4ccc(OCc5ccccc5)cc4=O)ccc32)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 14/20 0.58
KCNH2 Q12809 5/20 0.55
CYP3A4 P08684 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4444404 0.90 MCHR1 (0.52) MCHR1KCNH2CYP3A4
SCHEMBL4442735 0.88 MCHR1 (0.51) MCHR1KCNH2CYP3A4
SCHEMBL2891165 0.73 MCHR1 (1.00) MCHR1KCNH2
SCHEMBL4457815 0.73 MCHR1 (0.50) MCHR1
SCHEMBL1753898 0.73 MCHR1 (0.54) MCHR1KCNH2CYP3A4
SCHEMBL1005412 0.72 MCHR1 (1.00) MCHR1CYP3A4
Hydrochloric Acid SCHEMBL1003922 0.72 MCHR1 (0.98) MCHR1CYP3A4
SCHEMBL18154549 0.72 MCHR1 (0.61) MCHR1KCNH2CYP3A4
SCHEMBL10059384 0.71 MCHR1 (0.70) MCHR1KCNH2
SCHEMBL4881868 0.71 MCHR1 (0.71) MCHR1KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137270-A2 AZETIDINE DERIVATIVES H. LUNDBECK A/S (DK) 2009-11-12 WO disclosed