SCHEMBL13624159

SCHEMBL13624159

O=C(Cc1ccc(Cl)c([N+](=O)[O-])c1)Nc1ccc2[nH]c(-c3cscn3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 4/20 0.46
MAPT P10636 5/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.41
POLB P06746 2/20 0.41
MAOB P27338 1/20 0.41
KDR P35968 2/20 0.40
METAP2 P50579 2/20 0.40
LMNA P02545 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4376348 0.87 METAP1 (0.57) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4371202 0.85 KDR (0.55) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4377644 0.85 METAP1 (0.54) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4368921 0.85 METAP1 (0.54) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4367576 0.83 METAP1 (0.49) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4370849 0.82 MEN1 (0.53) METAP1KMT2AMEN1POLBMAOB
SCHEMBL4372206 0.82 METAP1 (0.45) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4367763 0.81 KDR (0.55) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4363482 0.81 METAP1 (0.52) METAP1MAPTNPC1RAB9AKMT2A
SCHEMBL4368752 0.81 KDR (0.46) METAP1MAPTNPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622592-B2 Carbonylamino-benzimidazole derivatives as androgen receptor modulators MERCK & CO., INC. (US) 2009-11-24 US disclosed