SCHEMBL13626641

SCHEMBL13626641

CCN(c1cc(OC)ccc1[C@@H]1CCc2cc(O)ccc2C1)C(C)c1ccc(OCCN(C)C(C)C)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.47
ESR2 Q92731 1/20 0.47
DRD2 P14416 6/20 0.35
DRD3 P35462 6/20 0.35
CYP26A1 O43174 1/20 0.35
DRD4 P21917 3/20 0.32
ROCK2 O75116 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626639 0.94 ESR1 (0.47) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626640 0.93 ESR1 (0.46) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626660 0.92 ESR1 (0.45) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626637 0.92 ESR1 (0.45) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626642 0.92 ESR1 (0.45) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626643 0.91 ESR1 (0.44) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626655 0.89 ESR1 (0.43) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626584 0.89 ESR1 (0.56) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626585 0.89 ESR1 (0.49) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626658 0.89 ESR1 (0.44) ESR1ESR2DRD2DRD3CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612114-B2 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-11-03 US disclosed