SCHEMBL13628745

SCHEMBL13628745

Cc1ncc(-c2ncn[nH]2)s1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.46
NPSR1 Q6W5P4 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
IDO1 P14902 6/20 0.34
HCAR2 Q8TDS4 1/20 0.33
ENPP2 Q13822 1/20 0.33
KDM4E B2RXH2 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628716 0.77 COMT (0.36) COMTALDH1A1GAAIDO1ENPP2
SCHEMBL10442596 0.73 HCAR2 (0.46) NPSR1CYP11B1CYP11B2HCAR2
SCHEMBL13628736 0.72 NPSR1 (0.33) NPSR1CYP11B1CYP11B2HCAR2
SCHEMBL18410397 0.71 SMPD3 (0.38) NPSR1CYP11B1CYP11B2HCAR2
SCHEMBL3744556 0.68 IDO1 (0.50) COMTALDH1A1IDO1ENPP2KDM4E
SCHEMBL20175445 0.66 HCAR2 (0.40) NPSR1CYP11B1CYP11B2HCAR2KDM4E
SCHEMBL13628752 0.65 NPSR1 (0.34) NPSR1CYP11B1CYP11B2HCAR2
SCHEMBL17289787 0.63 ADORA2A (0.35)
SCHEMBL4031086 0.63 POLB (0.48) ALDH1A1GAAIDO1ENPP2KDM4E
SCHEMBL10442133 0.63 NPC1 (0.39) NPSR1CYP11B1CYP11B2ALDH1A1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed