SCHEMBL13636369

SCHEMBL13636369

C=C(N)c1ccc(C)c(N)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.61
MAPT P10636 3/20 0.61
ALDH1A1 P00352 3/20 0.48
CASP1 P29466 2/20 0.48
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
CYP3A4 P08684 4/20 0.45
TSHR P16473 3/20 0.42
MAPK1 P28482 2/20 0.42
LMNA P02545 2/20 0.38
NPC1 O15118 1/20 0.38
MITF O75030 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 3/20 0.37
F2 P00734 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12824890 0.84 PRSS1 (0.64) TDP1MAPTALDH1A1PRSS1PRSS2
SCHEMBL8860069 0.83 MAPT (0.61) TDP1MAPTALDH1A1CASP1PRSS1
SCHEMBL18866954 0.83 MAPT (0.61) TDP1MAPTALDH1A1CASP1PRSS1
SCHEMBL22905073 0.79 TDP1 (0.42) TDP1MAPTALDH1A1CASP1PRSS1
SCHEMBL23592021 0.78 TSHR (0.50) TDP1MAPTALDH1A1CASP1PRSS1
SCHEMBL13495684 0.78 TDP1 (0.61) TDP1MAPTALDH1A1CASP1PRSS1
SCHEMBL284729 0.78 TDP1 (0.73) TDP1MAPTALDH1A1CASP1PRSS1
SCHEMBL20836577 0.78 TDP1 (0.55) TDP1MAPTALDH1A1CASP1PRSS1
SCHEMBL18773955 0.77 HDAC1 (0.52) TDP1MAPTALDH1A1PRSS1PRSS2
SCHEMBL13783388 0.76 MAPT (0.76) TDP1MAPTALDH1A1CASP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242385-B1 CYTOKINE, ESPECIALLY TNF-ALPHA, INHIBITORS PHARMACOPEIA INC (US) 2009-11-25 EP disclosed