SCHEMBL13638288

SCHEMBL13638288

C=C1CC(Nc2nccc(-c3ccc([C@H]4C[C@@H]4C(C)(C)O)s3)n2)CC(C)(C)N1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.32
CDK4 P11802 3/20 0.32
CCNB1 P14635 3/20 0.32
CCNA2 P20248 3/20 0.32
CCND1 P24385 3/20 0.32
CDK2 P24941 3/20 0.32
CCNA1 P78396 3/20 0.32
MAPK9 P45984 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638667 1.00 CDK1 (0.32) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL4491170 0.87 KCNH2 (0.35) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL4484036 0.87 KCNH2 (0.35) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL13638461 0.85 AKT3 (0.32) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL13638663 0.84 IKBKB (0.34) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL13638458 0.82 IKBKB (0.36) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL13638455 0.81 MAPK9 (0.33) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL13638557 0.81 IKBKB (0.45) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL13638500 0.81 IKBKB (0.33) CDK1CDK4CCNB1CCNA2CCND1
SCHEMBL14612785 0.80 IKBKB (0.37) CDK1CDK4CCNB1CCNA2CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed