SCHEMBL13639761

SCHEMBL13639761

O=C(C(=O)N1CCN(C(=O)c2ccccc2)CC1)c1c[nH]c2c(-c3cccs3)ccnc12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.49
CYP2C19 P33261 5/20 0.46
CYP3A4 P08684 3/20 0.44
CYP2D6 P10635 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2B6 P20813 1/20 0.43
KCNH2 Q12809 1/20 0.43
GBA1 P04062 1/20 0.43
ABL1 P00519 4/20 0.40
BCR P11274 4/20 0.40
TACR3 P29371 1/20 0.38
PLAUR Q03405 1/20 0.38
SLC6A7 Q99884 1/20 0.37
ALDH1A1 P00352 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1763503 0.88 CYP2C9 (0.49) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL2629049 0.87 CYP2C19 (0.65) CYP2C9CYP2C19CYP3A4CYP2D6SLC6A7
SCHEMBL2633348 0.87 CYP2C19 (0.65) CYP2C9CYP2C19CYP3A4CYP2D6SLC6A7
SCHEMBL1763035 0.85 CYP2C9 (0.48) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL2629052 0.85 CYP2C9 (0.49) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL1763197 0.84 CYP2C9 (0.48) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL15346088 0.83 CYP2C9 (0.50) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL2629034 0.82 CYP2C9 (0.52) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL1763071 0.82 CYP2C9 (0.49) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL1764105 0.82 CYP2C9 (0.55) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363705-B9 COMPOSITION AND ANTIVIRAL ACTIVITY OF SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2012-11-07 EP disclosed