SCHEMBL13650680

SCHEMBL13650680

CCOc1c(COC(C)O)cnn1Cc1nc(-c2cccc(C(F)(F)F)c2)cs1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.39
ITGB3 P05106 8/20 0.38
ITGA2B P08514 8/20 0.38
ITGB2 P05107 2/20 0.38
ICAM1 P05362 2/20 0.38
ITGAL P20701 2/20 0.38
TRPA1 O75762 2/20 0.37
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
AR P10275 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
TRPV3 Q8NET8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1198946 0.81 KDM4E (0.47) ITGB3ITGA2BITGB2ICAM1ITGAL
SCHEMBL1198797 0.80 KDM4E (0.53) ITGB3ITGA2BITGB2ICAM1ITGAL
SCHEMBL1199217 0.73 KDM4E (0.61) ITGB3ITGA2BITGB2ICAM1ITGAL
SCHEMBL1197463 0.72 ITGB2 (0.52) ITGB3ITGA2BITGB2ICAM1ITGAL
SCHEMBL1198442 0.70 KDM4E (0.56) ITGB3ITGA2BITGB2ICAM1ITGAL
SCHEMBL13650613 0.70 AR (0.55) ADAM17ITGB2ICAM1ITGALALDH1A1
SCHEMBL1198067 0.70 KDM4E (0.49) ITGB3ITGA2BITGB2ICAM1ITGAL
SCHEMBL1198444 0.70 MAPT (0.48) ITGB2ICAM1ITGALTRPA1ALDH1A1
SCHEMBL1197814 0.70 MEN1 (0.48) ITGB2ICAM1ITGALALDH1A1KDM4E
SCHEMBL1198790 0.68 ITGB2 (0.45) ITGB3ITGA2BITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009123316-A1 HETEROCYCLIC DERIVATIVE AND USE THEREOF 武田薬品工業株式会社 (JP) 2009-10-08 WO disclosed