SCHEMBL13655773

SCHEMBL13655773

O=C1Nc2ccccc2CCN1C1CCC=CCC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 12/20 0.44
RAMP1 O60894 4/20 0.44
NPC1 O15118 1/20 0.44
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44
MAPT P10636 1/20 0.41
BRD4 O60885 1/20 0.41
CREBBP Q92793 1/20 0.41
CHRM2 P08172 1/20 0.38
CHRM3 P20309 1/20 0.38
AHR P35869 1/20 0.38
PDK2 Q15119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16313925 0.88 MAPT (0.47) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL30178303 0.85 HTR2C (0.49) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL651023 0.85 HTR2C (0.49) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL3278838 0.85 CALCRL (0.44) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL1700379 0.85 CHRM2 (0.50) CALCRLRAMP1NPC1MAPK13MAPK12
Hydrochloric Acid SCHEMBL1819629 0.84 HTR2C (0.48) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL12401887 0.84 CALCRL (0.46) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL15144550 0.84 CALCRL (0.48) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL4718744 0.83 CALCRL (0.45) CALCRLRAMP1NPC1MAPK13MAPK12
SCHEMBL4718740 0.82 CALCRL (0.44) CALCRLRAMP1NPC1MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108648-A1 Selected CGRP antagonists, method for their manufacture and use as medicines Boehringer Ingelheim International GmbH (DE) 2009-10-14 EP disclosed