SCHEMBL13660429

SCHEMBL13660429

CCc1nc(C(C)(C)C)c2sccc2n1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 12/20 0.54
ADORA1 P30542 11/20 0.54
ADORA2B P29275 2/20 0.54
ADORA3 P0DMS8 1/20 0.54
PDE4A P27815 6/20 0.49
PDE4B Q07343 6/20 0.49
PDE4C Q08493 6/20 0.49
PDE4D Q08499 6/20 0.49
PDE3B Q13370 5/20 0.49
PDE3A Q14432 5/20 0.49
PDE7A Q13946 1/20 0.40
ELANE P08246 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14513332 0.90 ADORA2A (0.51) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL3679965 0.79 ADORA2A (0.77) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL4715461 0.77 ADORA2A (0.62) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL10171315 0.77 ADORA2A (0.58) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL179279 0.77 ADORA2A (0.44) ADORA2AADORA1ADORA2BADORA3PDE7A
SCHEMBL24995357 0.77 ADORA2A (0.60) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL10139170 0.77 ADORA2A (0.58) ADORA2AADORA1ADORA2BADORA3PDE7A
SCHEMBL19261286 0.76 ADORA2A (0.42) ADORA2AADORA1ADORA2BADORA3PDE7A
SCHEMBL9381944 0.76 ADORA2A (0.56) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL8363046 0.76 ADORA2A (0.42) ADORA2AADORA1ADORA2BADORA3PDE7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601713-B2 Kinase inhibitors and their uses RIGEL PHARMACEUTICALS, INC. (US) 2009-10-13 US disclosed