SCHEMBL13675125

SCHEMBL13675125

CC(C)(C)OC(=O)N1C[C@@H](NOCc2ccc(Cl)s2)CC1C(=O)Nc1ccc(N2CCOCC2=O)cc1C#N

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F10 P00742 19/20 0.39
F2 P00734 2/20 0.36
ABCB11 O95342 1/20 0.36
ST14 Q9Y5Y6 1/20 0.36
CYP1A2 P05177 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13672294 0.87 F10 (0.42) F10F2ABCB11ST14CYP3A4
SCHEMBL4484924 0.87 F10 (0.42) F10F2ABCB11ST14CYP3A4
SCHEMBL4484919 0.87 F10 (0.42) F10F2ABCB11ST14CYP3A4
SCHEMBL4479109 0.75 F10 (0.47) F10F2ABCB11ST14CYP3A4
SCHEMBL13672264 0.74 F10 (0.54) F10F2ABCB11ST14
SCHEMBL4485110 0.74 F10 (0.54) F10F2ABCB11ST14
SCHEMBL4485107 0.74 F10 (0.54) F10F2ABCB11ST14
SCHEMBL14534487 0.72 F10 (0.39) F10F2ABCB11ST14CYP1A2
SCHEMBL4492159 0.71 F10 (0.53) F10
SCHEMBL4492161 0.71 F10 (0.53) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601752-B2 Pyrrolidine derivatives HOFFMANN-LA ROCHE INC. (US) 2009-10-13 US disclosed