SCHEMBL13675158

SCHEMBL13675158

Cc1cc(Nc2ncnc3nc(Nc4ccc(CN5CCCC5)cc4)sc23)ccc1F

nearest known ligand 0.81

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.81
AXL P30530 1/20 0.45
CDK1 P06493 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13674980 0.99 EGFR (0.82) EGFRAXLCDK1
SCHEMBL13675194 0.93 EGFR (0.70) EGFRAXLCDK1
SCHEMBL13674979 0.93 EGFR (0.70) EGFRAXL
SCHEMBL13675161 0.92 EGFR (0.82) EGFRAXL
SCHEMBL13672611 0.90 EGFR (1.00) EGFRAXL
SCHEMBL13672599 0.89 EGFR (1.00) EGFRAXL
SCHEMBL13672615 0.89 EGFR (1.00) EGFRAXL
SCHEMBL13675193 0.89 EGFR (0.65) EGFRAXL
SCHEMBL14462155 0.87 EGFR (0.79) EGFRCDK1
SCHEMBL14461351 0.86 EGFR (0.79) EGFRCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7605154-B2 ATP-protein kinase inhibitors; cytomegalovirus; contraceptive agents; cancer; N7-(3-ethynyl-phenyl)-N2-(4-piperidin-1-ylmethyl-phenyl)-thiazolo[4,5-d]pyrimidine-2,7-diamine JANSSEN PHARMACEUTICA N.V. (BE) 2009-10-20 US disclosed