SCHEMBL13680357

SCHEMBL13680357

COc1cc2nc(C3(NC(=O)c4ccc5c(C6CCCC6)c(-c6ncc(Cl)cn6)n(C)c5c4)CCC3)n(C)c2cc1/C=C/C(C)=O

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2C8 P10632 1/20 0.56
CYP3A4 P08684 13/20 0.47
CYP2C19 P33261 12/20 0.47
HTR2A P28223 2/20 0.46
KCNH2 Q12809 1/20 0.44
SCN9A Q15858 2/20 0.40
CTSG P08311 1/20 0.39
MAOA P21397 1/20 0.39
DRD1 P21728 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680391 0.95 CYP2C9 (0.63) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL12899607 0.94 CYP1A2 (0.64) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL13680356 0.90 CYP1A2 (0.66) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL12899594 0.89 CYP1A2 (0.52) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL12899613 0.86 CYP3A4 (0.55) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL13680382 0.86 CYP1A2 (0.68) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL15109234 0.84 CYP1A2 (0.67) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL13680355 0.83 CYP1A2 (0.74) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL13680374 0.83 CYP1A2 (0.62) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19
SCHEMBL15109357 0.83 CYP1A2 (0.62) CYP2C9CYP1A2CYP2C8CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582770-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-09-01 US disclosed