SCHEMBL13686244

SCHEMBL13686244

Cc1ncccc1-c1cc(N2CCN(C)CC2)ncc1C(=O)N(C)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.81

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.81
GPBAR1 Q8TDU6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13686256 0.95 TACR1 (0.74) TACR1GPBAR1
SCHEMBL29467378 0.90 TACR1 (1.00) TACR1GPBAR1
SCHEMBL905330 0.90 TACR1 (1.00) TACR1GPBAR1
Hydrochloric Acid SCHEMBL905341 0.89 TACR1 (0.98) TACR1GPBAR1
SCHEMBL6637377 0.87 TACR1 (0.83) TACR1
SCHEMBL17762929 0.87 TACR1 (0.94) TACR1GPBAR1
Hydrochloric Acid SCHEMBL905337 0.87 TACR1 (0.81) TACR1
SCHEMBL6021041 0.86 TACR1 (0.78) TACR1
SCHEMBL3880526 0.86 TACR1 (0.61) TACR1GPBAR1
SCHEMBL17263543 0.86 TACR1 (0.92) TACR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856052-B1 NK1 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2009-09-02 EP disclosed
US-7176205-B2 Bi-pyridinyl derivatives as NK-1 antagonists HOFFMANN-LA ROCHE INC. (US) 2007-02-13 US disclosed
US-7176205-B2 Bi-pyridinyl derivatives as NK-1 antagonists HOFFMANN-LA ROCHE INC. (US) 2007-02-13 US disclosed