SCHEMBL13686649

SCHEMBL13686649

CCc1c(OC2CCN(C)CC2)ccc2cnccc12

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 5/20 0.43
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41
CHUK O15111 3/20 0.41
IGF1R P08069 1/20 0.38
TTK P33981 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
MELK Q14680 2/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
TLR9 Q9NR96 1/20 0.35
TLR7 Q9NYK1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12192620 0.84 IKBKB (0.51) IKBKBROCK2ROCK1CHUKMELK
SCHEMBL1706006 0.84 IKBKB (0.37) IKBKBROCK2ROCK1CHUK
SCHEMBL1706007 0.84 IKBKB (0.37) IKBKBROCK2ROCK1CHUK
SCHEMBL13686761 0.81 IKBKB (0.40) IKBKBROCK2ROCK1CHUKIGF1R
SCHEMBL12192784 0.76 IKBKB (0.50) IKBKBROCK2ROCK1CHUKMELK
Trifluoroacetic Acid SCHEMBL2496666 0.75 IKBKB (0.43) IKBKBROCK1CHUK
SCHEMBL13686654 0.73 LCK (0.43) IKBKBCHUKIGF1RTTKDYRK1B
SCHEMBL12192917 0.71 IKBKB (0.60) IKBKBROCK2ROCK1CHUKIGF1R
SCHEMBL15784007 0.71 ATR (0.45) IKBKBMELK
SCHEMBL13686682 0.70 IKBKB (0.54) IKBKBROCK1CHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899322-B1 ISOQUINOLINE DERIVATIVES AS INHIBITORS OF RHO-KINASE SANOFI AVENTIS (FR) 2009-09-02 EP disclosed