SCHEMBL1368665

SCHEMBL1368665

COc1cc(NC(=O)c2cccc(C(N)=O)c2-c2cnc3[nH]ccc3c2)cc(OC)c1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 2/20 0.56
BRD4 O60885 1/20 0.54
CDK8 P49336 7/20 0.47
CDK7 P50613 2/20 0.47
CCNT1 O60563 1/20 0.47
CCND1 P24385 1/20 0.47
CCNC P24863 1/20 0.47
CDK9 P50750 1/20 0.47
CCNH P51946 1/20 0.47
MNAT1 P51948 1/20 0.47
CDK6 Q00534 1/20 0.47
HTT P42858 1/20 0.47
PIK3CA P42336 1/20 0.45
MTOR P42345 1/20 0.45
RIPK1 Q13546 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
TOP1 P11387 1/20 0.43
PARP1 P09874 1/20 0.43
KDM4E B2RXH2 1/20 0.43
PLK4 O00444 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1368343 0.78 CDK8 (0.47) TNIKCDK8CDK7CCNT1CCND1
SCHEMBL1365527 0.74 TNIK (0.49) TNIKCDK8CDK7CCNT1CCND1
SCHEMBL4503280 0.74 P4HTM (0.52) TNIKBRD4PIK3CAMTORSMN1; SMN2
Hydrochloric Acid SCHEMBL1369411 0.73 TNIK (0.49) TNIKCDK8CDK7CCNT1CCND1
SCHEMBL29072615 0.73 TNIK (0.57) TNIKBRD4CDK8CDK7PIK3CA
SCHEMBL30580391 0.73 TNIK (0.57) TNIKBRD4CDK8CDK7PIK3CA
SCHEMBL720887 0.72 BRD4 (1.00) TNIKBRD4CDK8PIK3CARIPK1
SCHEMBL29072546 0.71 TNIK (0.57) TNIKBRD4CDK8CDK7CCNT1
SCHEMBL30580401 0.71 TNIK (0.57) TNIKBRD4CDK8CDK7CCNT1
SCHEMBL1368092 0.71 PIK3CA (0.48) TNIKBRD4CDK8CDK7CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067599-B2 Imidazo [4,5-B] pyridine and pyrrolo [2,3-B] pyridine protein kinase inhibitors HOFFMAN-LA ROCHE INC. (US) 2011-11-29 US claimed
US-8067599-B2 Imidazo [4,5-B] pyridine and pyrrolo [2,3-B] pyridine protein kinase inhibitors HOFFMAN-LA ROCHE INC. (US) 2011-11-29 US disclosed