SCHEMBL13688043

SCHEMBL13688043

Nc1ccc2c(c1)nc(Nc1ccc(F)c(Cl)c1)c1cscc12

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.54
CSNK2A1 P68400 8/20 0.49
CSNK2A2 P19784 2/20 0.49
CSNK2B P67870 2/20 0.49
ABCG2 Q9UNQ0 1/20 0.47
GRM1 Q13255 1/20 0.46
KDR P35968 1/20 0.44
MAPK1 P28482 1/20 0.43
BRAF P15056 1/20 0.43
SOS1 Q07889 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11932661 0.86 CSNK2A1 (0.45) EGFRCSNK2A1CSNK2A2CSNK2BABCG2
SCHEMBL13688023 0.85 CSNK2A1 (0.44) EGFRCSNK2A1CSNK2A2CSNK2BABCG2
SCHEMBL10134763 0.84 CSNK2A1 (0.46) EGFRCSNK2A1CSNK2A2CSNK2BABCG2
SCHEMBL13688029 0.83 EGFR (0.58) EGFRCSNK2A1CSNK2A2CSNK2BABCG2
SCHEMBL13688025 0.81 EGFR (0.60) EGFRCSNK2A1CSNK2A2CSNK2BABCG2
SCHEMBL10134772 0.79 CSNK2A1 (0.51) EGFRCSNK2A1CSNK2A2CSNK2BABCG2
SCHEMBL13688039 0.75 EGFR (0.61) EGFRCSNK2A1CSNK2A2CSNK2BABCG2
SCHEMBL13688035 0.72 MDM4 (0.42) EGFRKDR
SCHEMBL29923578 0.70 EGFR (1.00) EGFRGRM1KDRBRAF
SCHEMBL31299934 0.70 EGFR (1.00) EGFRGRM1KDRBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090239859-A1 PROTEIN KINASE MODULATORS SENHWA BIOSCIENCES, INC. (TW) 2009-09-24 US disclosed
WO-2009108912-A1 PROTEIN KINASE MODULATORS CYLENE PHARMACEUTICALS, INC. (US) 2009-09-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090239859-A1 PROTEIN KINASE MODULATORS PIM1, PIM2, PIM3 EGFR 580/4885CSNK2A1 680/4885CSNK2A2 810/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.