SCHEMBL13690909

SCHEMBL13690909

CCCCNc1ccc2c(COc3ccc(Cl)c(Oc4cc(Cl)cc(C#N)c4)c3)n[nH]c2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.43
CYP3A4 P08684 3/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
SLC22A12 Q96S37 1/20 0.33
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
ABCB1 P08183 1/20 0.30
ABCG2 Q9UNQ0 1/20 0.30
TBXA2R P21731 1/20 0.30
EGLN2 Q96KS0 1/20 0.30
EGLN1 Q9GZT9 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13690733 0.88 CYP3A4 (0.43) KCNH2CYP3A4CYP2D6CYP2C9CYP11B1
SCHEMBL3155350 0.88 CYP3A4 (0.41) KCNH2CYP3A4CYP2D6CYP2C9SLC22A12
SCHEMBL13119805 0.86 KCNH2 (0.48) KCNH2CYP3A4CYP2D6CYP2C9CYP11B1
SCHEMBL3159602 0.84 CYP3A4 (0.49) KCNH2CYP3A4CYP2D6CYP2C9CYP11B1
SCHEMBL3151052 0.84 CYP3A4 (0.55) KCNH2CYP3A4CYP2D6CYP2C9CYP11B1
SCHEMBL3145181 0.81 CYP3A4 (0.43) KCNH2CYP3A4CYP2D6CYP2C9CYP11B1
SCHEMBL30601611 0.81 KCNH2 (0.45) KCNH2CYP3A4CYP2D6CYP2C9CYP11B1
SCHEMBL3151001 0.81 KCNH2 (0.45) KCNH2CYP3A4CYP2D6CYP2C9CYP11B1
SCHEMBL3152053 0.80 CYP3A4 (0.42) KCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL3164134 0.79 CYP3A4 (0.42) KCNH2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009117278-A2 PROCESSES FOR PREPARING (AMINO-PYRAZOLOPYRIDINYL)METHOXY SUBSTITUTED BIARYL ETHERS MERCK & CO., INC. (US) 2009-09-24 WO disclosed