SCHEMBL13713009

SCHEMBL13713009

Nc1c(Br)cc(CC(NC(=O)N2CCC(N3CCc4ccccc4NC3=O)CC2)C(=O)N2CCC(N3CCCCC3)CC2)cc1C(F)(F)F

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 19/20 0.63
CYP3A4 P08684 16/20 0.63
RAMP1 O60894 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13331851 1.00 CALCRL (0.63) CALCRLCYP3A4RAMP1
SCHEMBL13331862 0.99 CALCRL (0.62) CALCRLCYP3A4RAMP1
SCHEMBL13713280 0.99 CALCRL (0.62) CALCRLCYP3A4RAMP1
SCHEMBL3313701 0.96 CALCRL (0.62) CALCRLCYP3A4RAMP1
SCHEMBL13331689 0.95 CALCRL (0.62) CALCRLCYP3A4RAMP1
SCHEMBL13713221 0.94 CALCRL (0.58) CALCRLCYP3A4RAMP1
SCHEMBL13331858 0.94 CALCRL (0.58) CALCRLCYP3A4RAMP1
SCHEMBL13331853 0.94 CALCRL (0.67) CALCRLCYP3A4RAMP1
SCHEMBL13713338 0.94 CALCRL (0.67) CALCRLCYP3A4RAMP1
SCHEMBL4361175 0.94 CALCRL (0.70) CALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7595312-B2 Selected CGRP antagonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2009-09-29 US disclosed