SCHEMBL13715575

SCHEMBL13715575

CCC(C)Oc1cc(N2CCN(C(=O)Cn3nc(C(F)(F)F)c(Cl)c3C)CC2)ccc1Cl

nearest known ligand 0.86

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 20/20 0.86
CYP2C19 P33261 1/20 0.78
KCNH2 Q12809 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2876791 0.92 CCR1 (1.00) CCR1CYP2C19KCNH2
SCHEMBL2866562 0.88 CCR1 (1.00) CCR1CYP2C19KCNH2
SCHEMBL2866978 0.88 CCR1 (1.00) CCR1CYP2C19KCNH2
SCHEMBL2874768 0.85 CCR1 (0.87) CCR1CYP2C19KCNH2
SCHEMBL13162691 0.85 CCR1 (0.93) CCR1CYP2C19KCNH2
SCHEMBL2875774 0.84 CCR1 (0.86) CCR1CYP2C19KCNH2
SCHEMBL2875657 0.84 CCR1 (0.82) CCR1CYP2C19KCNH2
SCHEMBL2869925 0.84 CCR1 (1.00) CCR1CYP2C19KCNH2
SCHEMBL13066146 0.84 CCR1 (0.78) CCR1CYP2C19KCNH2
SCHEMBL2866838 0.83 CCR1 (0.79) CCR1CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1531822-B1 1-ARYL-4-SUBSTITUTED PIPERAZINE DERIVATIVES FOR USE AS CCR1 ANTAGONISTS FOR THE TREATMENT OF INFLAMMATION AND IMMUNE DISORDERS CHEMOCENTRYX INC (US) 2009-08-05 EP disclosed