SCHEMBL13749604

SCHEMBL13749604

CNc1ncc(-c2ccnc(N)c2)cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.60
DYRK1A Q13627 4/20 0.49
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
IKBKE Q14164 1/20 0.43
TBK1 Q9UHD2 1/20 0.43
NOS3 P29474 3/20 0.42
NOS1 P29475 3/20 0.42
NOS2 P35228 3/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
FEN1 P39748 2/20 0.41
PDPK1 O15530 1/20 0.41
DHFR P00374 1/20 0.40
MAPT P10636 1/20 0.40
KHK P50053 1/20 0.38
AAK1 Q2M2I8 1/20 0.38
ROCK1 Q13464 1/20 0.38
CIT O14578 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30935767 0.78 DYRK1A (0.63) DYRK1AMKNK1MKNK2NOS3NOS1
SCHEMBL4402187 0.78 DYRK1A (0.63) DYRK1AMKNK1MKNK2NOS3NOS1
SCHEMBL8319877 0.78 DYRK1A (0.51) DYRK1AMKNK1MKNK2IKBKETBK1
Hydrochloric Acid SCHEMBL10461111 0.76 DYRK1A (0.61) DYRK1AMKNK1MKNK2NOS3NOS1
SCHEMBL17155080 0.76 DYRK1A (0.51) DYRK1AMKNK1MKNK2NOS3NOS1
SCHEMBL13633548 0.75 DYRK1A (0.62) MAP4K4DYRK1AMKNK1MKNK2NOS3
SCHEMBL4081141 0.75 DYRK1A (0.49) DYRK1AMKNK1MKNK2NOS3NOS1
SCHEMBL10918882 0.75 MAP4K4 (0.50) MAP4K4DYRK1AKDM4EMAPT
SCHEMBL30337203 0.74 DYRK1A (0.70) DYRK1AMKNK1MKNK2NOS3NOS1
SCHEMBL4619570 0.73 MAP4K4 (0.58) MAP4K4DYRK1AMKNK1MKNK2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737459-B1 IMIDAZOPYRIDINE AND IMIDAZOPYRIMIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS WARNER LAMBERT CO (US) 2009-08-05 EP disclosed