SCHEMBL13754152

SCHEMBL13754152

COc1ccc(-c2cc3c4c(c2)[C@@H]2CNCC[C@@H]2CN4CCC3)c(C(F)(F)F)c1

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.74
HTR2B P41595 9/20 0.74
HTR2A P28223 8/20 0.74
PROKR1 Q8TCW9 3/20 0.36
ESR1 P03372 1/20 0.35
EPHX2 P34913 1/20 0.34
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1E P28566 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
HTR7 P34969 1/20 0.34
HTR6 P50406 1/20 0.34
MAP4K1 Q92918 1/20 0.34
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3131164 1.00 HTR2C (0.74) HTR2CHTR2BHTR2APROKR1ESR1
SCHEMBL3134776 0.92 HTR2A (0.67) HTR2CHTR2BHTR2APROKR1ESR1
SCHEMBL3134771 0.92 HTR2A (0.67) HTR2CHTR2BHTR2APROKR1ESR1
SCHEMBL3136870 0.92 HTR2A (0.67) HTR2CHTR2BHTR2APROKR1ESR1
SCHEMBL3137627 0.88 HTR2A (0.61) HTR2CHTR2BHTR2APROKR1ESR1
SCHEMBL13268737 0.88 HTR2C (0.56) HTR2CHTR2BHTR2AESR1SIGMAR1
SCHEMBL5426076 0.85 HTR2C (1.00) HTR2CHTR2BHTR2AESR1EPHX2
SCHEMBL5407337 0.83 HTR2C (0.93) HTR2CHTR2BHTR2AESR1HTR1A
SCHEMBL5407340 0.83 HTR2C (0.93) HTR2CHTR2BHTR2AESR1HTR1A
SCHEMBL5413099 0.83 HTR2C (0.95) HTR2CHTR2BHTR2AESR1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399445-B1 SUBSTITUTED PYRROLOQUINOLINES AND PYRIDOQUINOLINES AS SEROTONIN AGONISTS AND ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2009-08-05 EP disclosed