SCHEMBL1375644

SCHEMBL1375644

CSc1ccc(CNc2n[nH]c3c(F)c(Cl)c(-c4ccccc4)cc23)cc1.Fc1cc(CNc2n[nH]c3c(F)c(Cl)c(-c4ccccc4)cc23)ccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.52
CDK1 P06493 2/20 0.52
CDK2 P24941 2/20 0.52
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 1/20 0.37
MAPK8 P45983 5/20 0.35
MAPK10 P53779 5/20 0.35
GRM4 Q14833 1/20 0.35
TGFBR1 P36897 1/20 0.34
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
FFAR1 O14842 1/20 0.34
RECQL P46063 1/20 0.34
MAP2K4 P45985 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2335590 0.93 GSK3B (0.58) GSK3BCDK1CDK2MEN1KMT2A
SCHEMBL2336401 0.92 GSK3B (0.58) GSK3BCDK1CDK2MEN1KMT2A
SCHEMBL6530031 0.84 GSK3B (0.50) GSK3BCDK1CDK2MAPK8MAPK10
SCHEMBL2338045 0.83 GSK3B (0.62) GSK3BCDK1CDK2MEN1KMT2A
SCHEMBL1375621 0.83 GSK3B (0.64) GSK3BCDK1CDK2MEN1KMT2A
SCHEMBL2360847 0.82 GSK3B (0.61) GSK3BCDK1CDK2MEN1KMT2A
SCHEMBL1378926 0.82 GSK3B (0.61) GSK3BCDK1CDK2MEN1KMT2A
SCHEMBL2335712 0.80 GSK3B (0.58) GSK3BCDK1CDK2MEN1KMT2A
SCHEMBL2336207 0.80 GSK3B (0.58) GSK3BCDK1CDK2MAPK8MAPK10
SCHEMBL6528915 0.79 GSK3B (0.57) GSK3BCDK1CDK2CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4764168-B2 2011-08-31 JP claimed