SCHEMBL13760880

SCHEMBL13760880

CCc1nc2c(cnn2CC)c(NC2CCOCC2)c1CNC(=O)c1cccc(C(=O)NCc2cccc(-c3cccc(CN4CCN(C(=O)OC(C)(C)C)C(C)C4)c3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 10/20 0.44
CHRM3 P20309 9/20 0.37
ROCK2 O75116 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1363909 1.00 PDE4B (0.44) PDE4BCHRM3ROCK2CHRM2CHRM1
SCHEMBL1363440 0.96 PDE4B (0.43) PDE4BCHRM3ROCK2
SCHEMBL1365292 0.95 PDE4B (0.41) PDE4BCHRM3ROCK2CHRM2CHRM1
SCHEMBL1362849 0.95 PDE4B (0.41) PDE4BCHRM3ROCK2
SCHEMBL1363194 0.94 CHRM3 (0.46) PDE4BCHRM3CHRM2CHRM1
SCHEMBL13750901 0.93 PDE4B (0.42) PDE4BROCK2
SCHEMBL13761019 0.93 PDE4B (0.42) PDE4BROCK2
SCHEMBL1362398 0.93 PDE4B (0.46) PDE4BCHRM3
SCHEMBL1364272 0.92 PDE4B (0.39) PDE4BCHRM3CHRM2CHRM1
SCHEMBL3425104 0.92 PDE4B (0.48) PDE4BCHRM3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100168-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed