SCHEMBL13765620

SCHEMBL13765620

CC(C)Oc1ccc(-c2nc(-c3ccc4c(c3)CCCN(C(=O)OC(C)(C)C)C4)no2)cc1N

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 18/20 0.49
S1PR3 Q99500 8/20 0.49
KCNH2 Q12809 2/20 0.48
ESR2 Q92731 1/20 0.41
NR1H2 P55055 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2989163 0.91 S1PR1 (0.60) S1PR1S1PR3KCNH2
SCHEMBL2993433 0.88 S1PR1 (0.65) S1PR1S1PR3KCNH2
SCHEMBL2605769 0.84 S1PR1 (0.56) S1PR1S1PR3KCNH2NR1H2
SCHEMBL13323054 0.83 S1PR1 (0.57) S1PR1S1PR3
SCHEMBL1966833 0.82 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL2605716 0.82 S1PR1 (0.63) S1PR1S1PR3KCNH2
SCHEMBL2605648 0.81 S1PR1 (0.47) S1PR1S1PR3KCNH2NR1H2
SCHEMBL2997333 0.80 S1PR1 (0.69) S1PR1S1PR3KCNH2
SCHEMBL13012428 0.80 S1PR1 (0.54) S1PR1S1PR3KCNH2
SCHEMBL2985518 0.79 S1PR1 (0.54) S1PR1S1PR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080725-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (SIP) GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed