SCHEMBL13765638

SCHEMBL13765638

O=CCN1CCc2ccc(-c3noc(-c4ccc(-c5ccccc5)c(C(F)(F)F)c4)n3)cc2CC1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.61
S1PR3 Q99500 6/20 0.55
S1PR4 O95977 1/20 0.43
CYP2C9 P11712 1/20 0.43
S1PR5 Q9H228 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10458912 0.90 S1PR1 (0.58) S1PR1S1PR3
SCHEMBL2983038 0.88 S1PR1 (0.75) S1PR1S1PR3
SCHEMBL2983598 0.84 S1PR1 (0.69) S1PR1S1PR3S1PR4CYP2C9S1PR5
Hydrochloric Acid SCHEMBL2986372 0.84 S1PR1 (0.68) S1PR1S1PR3S1PR4CYP2C9S1PR5
SCHEMBL2168613 0.83 S1PR1 (0.84) S1PR1S1PR3S1PR5
SCHEMBL2179933 0.83 S1PR1 (0.79) S1PR1S1PR3S1PR4CYP2C9S1PR5
SCHEMBL2181741 0.83 S1PR1 (0.79) S1PR1S1PR3S1PR4CYP2C9S1PR5
SCHEMBL10455382 0.82 S1PR1 (0.66) S1PR1S1PR3
SCHEMBL13765561 0.82 S1PR1 (0.57) S1PR1S1PR3S1PR5
SCHEMBL3068298 0.81 S1PR1 (0.63) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080725-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (SIP) GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed