SCHEMBL13769237

SCHEMBL13769237

C[C@@H]1CN(C(=O)OCc2ccccc2)CC1(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
HTR2C P28335 2/20 0.51
RORC P51449 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CYP2C19 P33261 1/20 0.50
HTT P42858 1/20 0.46
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45
PDK4 Q16654 1/20 0.45
CACNA1G O43497 1/20 0.45
CACNA1H O95180 1/20 0.45
CACNA1I Q9P0X4 1/20 0.45
ALDH1A1 P00352 1/20 0.44
CTSK P43235 1/20 0.43
GRIN2B Q13224 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12167420 1.00 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL4174274 0.87 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL4181131 0.87 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL4174279 0.87 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL1189044 0.86 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL12492571 0.86 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL12167385 0.86 SMN1; SMN2 (0.49) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL1189001 0.85 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL12683506 0.85 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AHTR2CRORC
SCHEMBL15883700 0.85 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9AHTR2CRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7563805-B2 7-[3-Amino-3,4-dimethylpyrrolidine-1-yl]-6-fluoro-1-[(1R,2S)-2-fluorocyclopropyl]-1,4-dihydro-8-methyl-4-oxoquinoline-3-carboxylic acid: quinoline bactericide; broad spectrum, strong antibacterial activity for Grampositive/-negative including multiple resistant cocci; side effect reductcion; drug design DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2009-07-21 US disclosed