SCHEMBL13769259

SCHEMBL13769259

COC(=O)COc1nc(C2CC2)nc(C)c1C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.42
MAPK1 P28482 2/20 0.38
ALDH1A1 P00352 2/20 0.37
PTGDR Q13258 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
PDE10A Q9Y233 4/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
LDHA P00338 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
KDM4E B2RXH2 2/20 0.32
GLA P06280 1/20 0.32
NR1I2 O75469 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL718535 0.93 TSHR (0.41) TSHRMAPK1ALDH1A1PTGDRPTGDR2
SCHEMBL717059 0.87 TSHR (0.38) TSHRMAPK1ALDH1A1PTGDRPTGDR2
SCHEMBL718995 0.86 PDE10A (0.50) PTGDRPTGDR2PDE10ANR1I2CYP3A4
SCHEMBL719801 0.86 PDE10A (0.44) TSHRMAPK1ALDH1A1PTGDRPTGDR2
SCHEMBL1609158 0.81 PDE10A (0.39) TSHRMAPK1ALDH1A1PDE10ANR1I2
SCHEMBL718722 0.77 ALOX5AP (0.36) TSHRMAPK1ALDH1A1PDE10AKMT2A
SCHEMBL721836 0.71 PDE10A (0.53) PDE10ANR1I2CYP3A4CYP2D6
SCHEMBL12713482 0.70 SYK (0.36) PDE10ANR1I2CYP3A4CYP2D6
SCHEMBL14440830 0.68 PDE10A (0.58) PDE10A
SCHEMBL1609868 0.68 PDE10A (0.35) PDE10ANR1I2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081112-A2 CHEMICAL COMPOUNDS SYNGENTA LIMITED (GB) 2009-07-02 WO disclosed