SCHEMBL13769445

SCHEMBL13769445

CBC(C)(C(=O)NC1CCN(c2nc(-c3ccccc3O)nc3ccccc23)CC1)C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMAD3 P84022 1/20 0.53
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
CHEK2 O96017 6/20 0.52
TSHR P16473 5/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HIF1A Q16665 2/20 0.44
CYP1A2 P05177 4/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 3/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPK1 P28482 1/20 0.43
TP53 P04637 2/20 0.43
CLK4 Q9HAZ1 2/20 0.41
USP2 O75604 2/20 0.41
ALOX15 P16050 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSP90AA1 P07900 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1622626 0.89 SMAD3 (0.55) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL1624268 0.86 SMAD3 (0.59) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL1624722 0.83 SMAD3 (0.55) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL13769806 0.82 SMAD3 (0.54) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL1623313 0.82 SMAD3 (0.67) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL1621972 0.82 SMAD3 (0.56) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL1624000 0.81 SMAD3 (0.57) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL1623965 0.80 MEN1 (0.44) SMAD3MEN1KMT2ACHEK2TSHR
SCHEMBL13080749 0.77 TSHR (0.57) MEN1KMT2ATSHRALDH1A1MAPT
SCHEMBL1622627 0.77 MEN1 (0.47) SMAD3MEN1KMT2ACHEK2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed