SCHEMBL13769449

SCHEMBL13769449

C[C@H]1CCN(c2nc(-c3ccccc3O)nc3ccc(F)cc23)C1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 5/20 0.62
SMAD3 P84022 1/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
HIF1A Q16665 3/20 0.50
MAPT P10636 5/20 0.49
ALDH1A1 P00352 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
KDM4E B2RXH2 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
TSHR P16473 3/20 0.46
LMNA P02545 2/20 0.45
HTT P42858 2/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
TP53 P04637 3/20 0.43
USP2 O75604 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TLR7 Q9NYK1 1/20 0.42
ADORA2A P29274 1/20 0.41
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1084341 0.89 HIF1A (0.57) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL183923 0.88 CHEK2 (0.58) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL183922 0.88 CHEK2 (0.58) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL1084929 0.88 CHEK2 (0.56) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL1084555 0.88 CHEK2 (0.80) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL1084832 0.88 CHEK2 (0.80) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL1084343 0.87 CHEK2 (0.56) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL1084638 0.87 CHEK2 (0.56) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL1621893 0.86 SMAD3 (0.56) CHEK2SMAD3MEN1KMT2AHIF1A
SCHEMBL1623570 0.86 CHEK2 (0.55) CHEK2SMAD3MEN1KMT2AHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed