SCHEMBL13769476

SCHEMBL13769476

Cc1ccc2c(N3CCN(C(=O)CCC(C)(C)C)CC3)nc(-c3c(O)cccc3F)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.43
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
KRAS P01116 5/20 0.37
MAPT P10636 2/20 0.37
HRH4 Q9H3N8 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
EGFR P00533 1/20 0.36
HMOX2 P30519 1/20 0.36
CRYZ Q08257 1/20 0.36
VAT1 Q99536 1/20 0.36
RTN4 Q9NQC3 1/20 0.36
CHRM1 P11229 1/20 0.36
PARP1 P09874 1/20 0.35
GBA1 P04062 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1623848 0.85 CHEK2 (0.42) CHEK2LMNATP53KRASMAPT
SCHEMBL13568165 0.85 CHEK2 (0.42) CHEK2LMNATP53KRASMAPT
SCHEMBL1623851 0.85 CHEK2 (0.42) CHEK2LMNATP53KRASMAPT
Hydrochloric Acid SCHEMBL1622281 0.84 CHEK2 (0.42) CHEK2LMNATP53KRASMAPT
Hydrochloric Acid SCHEMBL1622285 0.84 CHEK2 (0.42) CHEK2LMNATP53KRASMAPT
SCHEMBL1084945 0.84 MEN1 (0.51) CHEK2LMNAMAPTMEN1KMT2A
SCHEMBL1622534 0.84 CHEK2 (0.44) CHEK2KRASMAPTHRH4MEN1
SCHEMBL13079915 0.84 CHEK2 (0.44) CHEK2KRASMAPTHRH4MEN1
SCHEMBL1622531 0.84 CHEK2 (0.44) CHEK2KRASMAPTHRH4MEN1
SCHEMBL13769484 0.82 HRH4 (0.55) CHEK2LMNAMAPTHRH4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed