SCHEMBL13769717

SCHEMBL13769717

CC1CCC(C)N1c1ncnc2c1c(-c1cccc(Cl)c1Cl)cn2CC(=O)N1CCC(n2c(=O)[nH]c3ncccc32)CC1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 19/20 0.55
PIK3CD O00329 1/20 0.44
PDE2A O00408 1/20 0.44
PDE4A P27815 1/20 0.44
PIK3R1 P27986 1/20 0.44
PIK3CA P42336 1/20 0.44
PDE1A P54750 1/20 0.44
PDE1B Q01064 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE1C Q14123 1/20 0.44
PDE3A Q14432 1/20 0.44
PDE10A Q9Y233 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13770230 0.90 CALCRL (0.58) CALCRL
SCHEMBL4007941 0.90 CALCRL (0.60) CALCRL
SCHEMBL13769990 0.89 CALCRL (0.57) CALCRLPIK3CDPDE2APDE4APIK3R1
SCHEMBL13769779 0.89 CALCRL (0.56) CALCRLPIK3CDPDE2APDE4APIK3R1
SCHEMBL13770231 0.89 CALCRL (0.57) CALCRL
SCHEMBL13769985 0.88 CALCRL (0.54) CALCRLPIK3CDPDE2APDE4APIK3R1
SCHEMBL4012303 0.88 CALCRL (0.58) CALCRL
SCHEMBL4012312 0.87 CALCRL (0.56) CALCRL
SCHEMBL13769716 0.87 CALCRL (0.56) CALCRL
SCHEMBL13770229 0.86 CALCRL (0.56) CALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed