SCHEMBL13786147

SCHEMBL13786147

CCc1cc(C(CC)(CC)c2ccc(S(=O)(=O)NCC(=O)OC)s2)ccc1OCC(N=O)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 10/20 0.35
HDAC3 O15379 6/20 0.35
HDAC1 Q13547 1/20 0.33
VDR P11473 5/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
AR P10275 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3389821 0.89 HDAC6 (0.46) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13786148 0.84 HDAC6 (0.42) HDAC6HDAC3HDAC1VDRAR
SCHEMBL3389811 0.84 HDAC6 (0.46) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13366712 0.82 PPARG (0.37) HDAC6HDAC3HDAC1VDRKDM4E
SCHEMBL3392979 0.81 HDAC6 (0.54) HDAC6HDAC3HDAC1VDRAR
SCHEMBL3388902 0.81 HDAC6 (0.46) HDAC6HDAC3HDAC1VDRAR
SCHEMBL13786313 0.81 HDAC6 (0.46) HDAC6HDAC3HDAC1VDRAR
SCHEMBL4421979 0.76 HDAC6 (0.46) HDAC6HDAC3HDAC1VDRAR
SCHEMBL3391254 0.74 HDAC6 (0.55) HDAC6HDAC3HDAC1VDRAR
Acetic Acid Methyl Ester SCHEMBL3389823 0.74 HDAC6 (0.47) HDAC6HDAC3HDAC1VDRAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511740-B1 PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS LILLY CO ELI (US) 2009-07-08 EP disclosed