SCHEMBL13786397

SCHEMBL13786397

CCCCOC(=O)CC1c2ccc(-c3noc(-c4ccc(OC(C)C)c(N)c4)n3)c(C)c2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.42
S1PR5 Q9H228 5/20 0.42
S1PR3 Q99500 4/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3755317 0.93 S1PR1 (0.48) S1PR1S1PR5S1PR3CYP3A4CYP2C9
SCHEMBL3752329 0.92 S1PR1 (0.53) S1PR1S1PR5S1PR3CYP3A4CYP2C9
SCHEMBL13786427 0.86 S1PR1 (0.49) S1PR1S1PR5S1PR3CYP3A4CYP2C9
SCHEMBL3750162 0.82 S1PR1 (0.56) S1PR1S1PR5S1PR3CYP2C9
SCHEMBL3758679 0.81 S1PR1 (0.61) S1PR1S1PR5S1PR3CYP3A4CYP2C9
SCHEMBL3749885 0.81 S1PR1 (0.49) S1PR1S1PR5S1PR3CYP3A4CYP2C9
SCHEMBL3757708 0.80 S1PR1 (0.55) S1PR1S1PR5S1PR3CYP3A4CYP2C9
SCHEMBL3661119 0.79 S1PR1 (0.56) S1PR1S1PR5S1PR3CYP2C9
SCHEMBL13012428 0.78 S1PR1 (0.54) S1PR1S1PR5S1PR3CYP3A4CYP2C9
SCHEMBL3658685 0.78 S1PR1 (0.61) S1PR1S1PR5S1PR3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080728-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (SIP) GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed