SCHEMBL13787103

SCHEMBL13787103

Bc1ccc2oc3c(=O)[nH]c(-c4ccc(NC(=O)c5ccc(OC)nc5)cc4Cl)nc3c2c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 19/20 0.53
CSNK2A2 P19784 19/20 0.53
CSNK2B P67870 19/20 0.53
PIM3 Q86V86 18/20 0.53
PIM2 Q9P1W9 18/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1854554 0.91 PIM1 (0.61) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL12661065 0.89 PIM1 (0.53) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1853836 0.85 CSNK2A2 (0.56) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL13787107 0.85 PIM1 (0.53) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL12660263 0.81 PIM1 (0.55) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL13787070 0.81 PIM1 (0.57) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1849067 0.81 PIM1 (0.63) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1849830 0.81 PIM1 (0.61) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1851723 0.80 PIM1 (0.64) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL1849522 0.80 PIM1 (0.62) PIM1CSNK2A2CSNK2BPIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009086264-A1 BENZOFUROPYRIMIDINONES AS PROTEIN KINASE INHIBITORS EXELIXIS, INC. (US) 2009-07-09 WO disclosed