SCHEMBL13798697

SCHEMBL13798697

CSc1nc(-c2cccc(O)c2)c2c(C#N)cn(COCC[Si](C)(C)C)c2n1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
HSP90AB1 P08238 1/20 0.35
LHCGR P22888 1/20 0.35
ADORA2A P29274 3/20 0.32
ADORA1 P30542 3/20 0.32
CYP19A1 P11511 1/20 0.32
ADORA2B P29275 1/20 0.32
AR P10275 1/20 0.31
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2565245 0.89 HSP90AB1 (0.41) CHUKHSP90AB1
SCHEMBL13798696 0.83 HSP90AB1 (0.40) HSP90AB1ADORA2AADORA1
SCHEMBL2567605 0.80 HSP90AB1 (0.52) HSP90AB1PDE10A
SCHEMBL13798694 0.78 HSP90AB1 (0.54) HSP90AB1
SCHEMBL3561868 0.78 LRRK2 (0.46) CYP19A1AR
SCHEMBL2562784 0.78 CYP1A2 (0.33) HSP90AB1
SCHEMBL2564812 0.77 KLKB1 (0.32)
SCHEMBL2568420 0.77 HSP90AB1 (0.47) HSP90AB1
SCHEMBL2566599 0.76 KCNH2 (0.43) HSP90AB1
SCHEMBL2565058 0.76 HSP90AB1 (0.46) HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090163490-A1 Pyrrolopyrimidine Derivatives Used As HSP90 Inhibitors VERNALIS (R&D) LTD. (GB) 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163490-A1 Pyrrolopyrimidine Derivatives Used As HSP90 Inhibitors HSP90AA1, HSP90AB1, RAF1 IKBKB 756/4885CHUK 258/4885HSP90AB1 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.