SCHEMBL13802157

SCHEMBL13802157

COCOc1ccc2sc(CSC(C)(C)C=O)cc2c1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.35
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CA2 P00918 2/20 0.32
F2RL3 Q96RI0 1/20 0.31
CLK1 P49759 1/20 0.30
DYRK1A Q13627 1/20 0.30
DYRK1B Q9Y463 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13791184 0.88 BACE1 (0.40) BACE1PDE3BPDE3ACA2F2RL3
SCHEMBL3907282 0.79 PPARA (0.36) BACE1CA2CLK1DYRK1ADYRK1B
SCHEMBL3914986 0.78 BACE1 (0.38) BACE1PDE3BPDE3ACA2F2RL3
SCHEMBL13802139 0.78 DYRK1A (0.42) CA2CLK1DYRK1ADYRK1B
SCHEMBL13790850 0.76 BACE1 (0.45) BACE1PDE3BPDE3ACA2F2RL3
SCHEMBL3905190 0.74 CYP2A6 (0.47) BACE1PDE3BPDE3ACA2F2RL3
SCHEMBL3903263 0.73 CYP2A6 (0.54) BACE1PDE3BPDE3ACA2F2RL3
SCHEMBL13802155 0.73 BACE1 (0.43) BACE1PDE3BPDE3ACA2F2RL3
SCHEMBL3911211 0.71 BACE1 (0.41) BACE1PDE3BPDE3ACA2F2RL3
SCHEMBL13791095 0.70 BACE1 (0.44) BACE1PDE3BPDE3ACA2F2RL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553867-B2 Furan or thiophene derivative and medicinal use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-30 US disclosed