SCHEMBL13809378

SCHEMBL13809378

O=C(NC1CCN(Cc2ccccc2)CC1)c1ccc2[nH]c3c(c2c1)CN(Cc1ccc(F)cc1)CC3

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.64
HDAC6 Q9UBN7 3/20 0.64
ACHE P22303 2/20 0.63
MCHR1 Q99705 3/20 0.62
SIGMAR1 Q99720 3/20 0.62
SLC6A12 P48065 2/20 0.62
TMEM97 Q5BJF2 1/20 0.62
AKR1B1 P15121 1/20 0.59
ROCK2 O75116 1/20 0.54
ROCK1 Q13464 1/20 0.54
TP53 P04637 1/20 0.53
DRD4 P21917 2/20 0.53
SLC6A13 Q9NSD5 1/20 0.53
DRD2 P14416 1/20 0.53
ATM Q13315 1/20 0.52
GPR55 Q9Y2T6 1/20 0.52
CCR3 P51677 1/20 0.52
HTR6 P50406 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL61297 0.93 HDAC1 (0.63) HDAC1HDAC6ACHEMCHR1SIGMAR1
SCHEMBL60695 0.92 HDAC1 (0.58) HDAC1HDAC6ACHEMCHR1SIGMAR1
SCHEMBL62174 0.91 HDAC1 (0.64) HDAC1HDAC6ACHEMCHR1SIGMAR1
SCHEMBL61826 0.91 DRD4 (0.61) HDAC1HDAC6ACHEMCHR1SIGMAR1
SCHEMBL61772 0.90 HDAC1 (0.61) HDAC1HDAC6ACHEMCHR1SIGMAR1
SCHEMBL61323 0.90 AKR1B1 (0.57) HDAC1HDAC6ACHESIGMAR1SLC6A12
SCHEMBL60899 0.90 AKR1B1 (0.56) HDAC1HDAC6ACHESLC6A12AKR1B1
SCHEMBL16927810 0.88 HDAC1 (0.57) HDAC1HDAC6ACHEMCHR1SIGMAR1
SCHEMBL61090 0.88 HDAC1 (0.58) HDAC1HDAC6ACHESLC6A12AKR1B1
SCHEMBL10168433 0.88 HDAC1 (0.61) HDAC1HDAC6ACHEMCHR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009076631-A1 CARBOXAMIDE, SULFONAMIDE AND AMINE COMPOUNDS FOR METABOLIC DISORDERS RIGEL PHARMACEUTICALS, INC. (US) 2009-06-18 WO disclosed