SCHEMBL13811530

SCHEMBL13811530

COc1cc(Cl)c(-c2nc(SC(C)C(=O)O)nc3c2C(C#N)CN3)cc1OCCN1CCC(F)(F)C1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 7/20 0.59
NSD2 O96028 2/20 0.38
KCNH2 Q12809 1/20 0.35
MCHR1 Q99705 1/20 0.35
HTR2C P28335 2/20 0.34
HTR2A P28223 1/20 0.34
HSP90AA1 P07900 1/20 0.32
PDGFRB P09619 2/20 0.32
ADAMTS5 Q9UNA0 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
EIF4EBP1 Q13541 1/20 0.31
CCNK O75909 1/20 0.31
CDK12 Q9NYV4 1/20 0.31
SRC P12931 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13811529 0.88 HSP90AB1 (0.54) HSP90AB1NSD2KCNH2HTR2CHTR2A
SCHEMBL12161032 0.81 HSP90AB1 (0.87) HSP90AB1NSD2KCNH2HSP90AA1SRC
SCHEMBL12161232 0.76 HSP90AB1 (0.84) HSP90AB1NSD2KCNH2HSP90AA1SRC
SCHEMBL13811528 0.74 HSP90AB1 (0.42) HSP90AB1NSD2MCHR1HTR2CHTR2A
SCHEMBL12161199 0.74 HSP90AB1 (1.00) HSP90AB1NSD2KCNH2HSP90AA1SRC
SCHEMBL2567990 0.73 HSP90AB1 (0.81) HSP90AB1KCNH2HSP90AA1SRC
SCHEMBL13811667 0.73 HSP90AB1 (0.62) HSP90AB1KCNH2HSP90AA1SRC
SCHEMBL12160986 0.72 HSP90AB1 (1.00) HSP90AB1NSD2KCNH2HSP90AA1
SCHEMBL2565203 0.70 HSP90AB1 (0.77) HSP90AB1KCNH2HSP90AA1SRC
SCHEMBL12161036 0.69 HSP90AB1 (0.92) HSP90AB1KCNH2HSP90AA1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090163490-A1 Pyrrolopyrimidine Derivatives Used As HSP90 Inhibitors VERNALIS (R&D) LTD. (GB) 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163490-A1 Pyrrolopyrimidine Derivatives Used As HSP90 Inhibitors HSP90AA1, HSP90AB1, RAF1 HSP90AB1 2/4885NSD2 2144/4885KCNH2 2202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.