SCHEMBL13818263

SCHEMBL13818263

O=C1COc2cc(F)c(F)cc2N1CCCN1C2CCC1CC(=CCOCC1CC1)C2

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 7/20 0.45
CHRM5 P08912 1/20 0.40
CHRM3 P20309 1/20 0.40
DRD2 P14416 7/20 0.34
KCNH2 Q12809 5/20 0.34
HTR2A P28223 2/20 0.33
MCHR1 Q99705 2/20 0.33
EGFR P00533 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13818261 0.90 CHRM1 (0.45) CHRM1CHRM5CHRM3DRD2KCNH2
SCHEMBL4098902 0.84 CHRM1 (0.44) CHRM1CHRM5CHRM3DRD2KCNH2
SCHEMBL4101713 0.81 CHRM1 (0.48) CHRM1CHRM5CHRM3DRD2KCNH2
SCHEMBL13818265 0.81 CHRM1 (0.48) CHRM1CHRM5CHRM3DRD2KCNH2
SCHEMBL13692826 0.75 CHRM1 (0.44) CHRM1CHRM5CHRM3DRD2KCNH2
SCHEMBL4089822 0.73 CHRM1 (0.60) CHRM1CHRM5CHRM3DRD2KCNH2
SCHEMBL15617903 0.72 CHRM1 (0.46) CHRM1CHRM5CHRM3DRD2KCNH2
SCHEMBL4103787 0.71 CHRM1 (0.42) CHRM1DRD2HTR2AMCHR1
SCHEMBL15589859 0.71 CHRM1 (0.42) CHRM1DRD2HTR2AMCHR1
SCHEMBL13692823 0.71 CHRM1 (0.42) CHRM1DRD2HTR2AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550459-B2 Neurodegenerative diseases, psychological disorders; e.g. 4-[3-(3a -Cyclopropylmethoxy-8-azabicyclo[3.2.1]oct-8-yl)-2-methylpropyl]-4H-benzo[1.4]oxazin-3-one ACADIA PHARMACEUTICALS, INC. (US) 2009-06-23 US disclosed
US-7550459-B2 Neurodegenerative diseases, psychological disorders; e.g. 4-[3-(3a -Cyclopropylmethoxy-8-azabicyclo[3.2.1]oct-8-yl)-2-methylpropyl]-4H-benzo[1.4]oxazin-3-one ACADIA PHARMACEUTICALS, INC. (US) 2009-06-23 US disclosed