SCHEMBL13824734

SCHEMBL13824734

Cc1csc(-c2ccc3c(n2)CC(C)(C)CC3=O)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.61
ALDH1A1 P00352 4/20 0.48
HTT P42858 2/20 0.48
RXFP1 Q9HBX9 1/20 0.41
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 1/20 0.40
GRM5 P41594 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PDE10A Q9Y233 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
POLB P06746 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13707014 0.86 CYP2C19 (0.52) CYP2C19ALDH1A1HTTRXFP1PIK3CD
SCHEMBL13707073 0.79 CYP2C19 (0.54) CYP2C19ALDH1A1HTTRXFP1PIK3CD
SCHEMBL13706972 0.78 GRM5 (0.41) ALDH1A1KDM4ENPC1GRM5RAB9A
SCHEMBL25717168 0.77 CYP2C19 (1.00) CYP2C19ALDH1A1HTTKDM4ENPC1
SCHEMBL13706911 0.75 GRM5 (0.45) CYP2C19ALDH1A1KDM4ENPC1GRM5
SCHEMBL4333936 0.75 CYP2C19 (0.56) CYP2C19ALDH1A1HTTKDM4ENPC1
SCHEMBL8284605 0.74 CYP2C19 (0.54) CYP2C19ALDH1A1HTTPIK3CDPIK3CA
SCHEMBL13824424 0.74 CYP2C19 (0.61) CYP2C19ALDH1A1HTTKDM4ENPC1
SCHEMBL13707029 0.73 CYP2C19 (0.50) CYP2C19ALDH1A1HTTRXFP1PIK3CD
SCHEMBL11644246 0.73 CYP2C19 (0.60) CYP2C19ALDH1A1HTTRXFP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550482-B2 Tetrahydroquinolones and their use as modulators of metabotropic glutamate receptors MERZ PHARMA GMBH & CO. KGAA (DE) 2009-06-23 US disclosed