SCHEMBL13825281

SCHEMBL13825281

Bc1nnc(SCC(=O)Nc2ccc(S(N)(=O)=O)cc2Cl)n1-c1ccc(C2CC2)c2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 16/20 0.54
SLC2A9 Q9NRM0 3/20 0.54
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
SLC22A11 Q9NSA0 1/20 0.47
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 1/20 0.45
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA5B Q9Y2D0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL247372 0.92 SLC22A12 (0.54) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL248867 0.91 SLC22A12 (0.66) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL30601618 0.91 SLC22A12 (0.66) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL3435532 0.91 SLC22A12 (0.54) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL3435725 0.89 SLC22A12 (0.52) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL1719905 0.82 SLC22A12 (0.55) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL249261 0.82 SLC22A12 (0.66) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL1720398 0.82 SLC22A12 (0.54) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL12011401 0.81 CA1 (0.46) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2
SCHEMBL843191 0.81 SLC22A12 (0.54) SLC22A12SLC2A9CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402011-B1 S-triazolyl alpha-mercaptoacetanilides as inhibitors of HIV reverse transcriptase ARDEA BIOSCIENCES INC (US) 2012-11-14 EP disclosed