SCHEMBL1384515

SCHEMBL1384515

Cn1c(CN2C(=O)CN(S(=O)(=O)C=Cc3ccc(Cl)s3)CC2CO)cc2cnccc21

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
F10 P00742 14/20 0.49
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27526785 0.90 F10 (0.48) F10CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4390586 0.87 F10 (0.44) F10
SCHEMBL4390583 0.87 F10 (0.44) F10
SCHEMBL1652716 0.82 F10 (0.70) F10CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1652862 0.82 F10 (0.70) F10CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1652714 0.82 F10 (0.70) F10CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1386589 0.78 F10 (0.71) F10
SCHEMBL4391897 0.78 F10 (0.41) F10
SCHEMBL4397921 0.76 F10 (0.44) F10CYP2C9
SCHEMBL4397916 0.76 F10 (0.44) F10CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4829449-B2 2011-12-07 JP claimed
JP-2003508353-A 2003-03-04 JP claimed
EP-1208097-A2 SUBSTITUTED OXOAZAHETEROCYCLYL COMPOUNDS Aventis Pharmaceuticals Inc. (US) 2002-05-29 EP claimed
WO-2001007436-A2 SUBSTITUTED OXOAZAHETEROCYCLYL COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2001-02-01 WO claimed