SCHEMBL13846558

SCHEMBL13846558

ONc1cnc(NCc2ccccc2OC(F)(F)F)cc1NCC1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
PRKCQ Q04759 6/20 0.43
PIM1 P11309 4/20 0.43
CHEK1 O14757 5/20 0.40
PRKCD Q05655 4/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
FLT3 P36888 3/20 0.38
KCNH2 Q12809 2/20 0.38
PIM3 Q86V86 2/20 0.38
PIM2 Q9P1W9 2/20 0.38
TACR1 P25103 1/20 0.38
CCNT1 O60563 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3984374 0.84 PRKCQ (0.58) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13846480 0.77 PRKCQ (0.51) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13620030 0.76 PRKCQ (0.49) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13846554 0.76 PRKCQ (0.62) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13846611 0.75 PRKCQ (0.60) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13846604 0.75 PRKCQ (0.60) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13846606 0.74 PRKCQ (0.51) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13846553 0.74 PRKCQ (0.60) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL13846563 0.74 PRKCQ (0.60) HDAC3HDAC1HDAC2HDAC6PRKCQ
SCHEMBL3986930 0.74 PRKCQ (0.72) PRKCQPIM1PRKCDPIM3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1866286-B1 PYRIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA BOEHRINGER INGELHEIM PHARMA (DE) 2009-05-27 EP disclosed