SCHEMBL13848902

SCHEMBL13848902

O=C(Nc1cccc(-c2cc(Cc3cc[n+]([O-])cc3)cc3cccnc23)c1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 11/20 0.54
PDE4B Q07343 9/20 0.54
PDE4C Q08493 8/20 0.54
PDE4D Q08499 8/20 0.54
GAA P10253 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CFD P00746 1/20 0.45
PABPC1 P11940 1/20 0.43
ENPP1 P22413 1/20 0.43
KDR P35968 1/20 0.43
KCNK3 O14649 1/20 0.43
KCNK9 Q9NPC2 1/20 0.43
KMT2A Q03164 1/20 0.42
PRKD3 O94806 1/20 0.41
ABL1 P00519 1/20 0.41
PRKCG P05129 1/20 0.41
PRKCB P05771 1/20 0.41
PDGFRB P09619 1/20 0.41
BCR P11274 1/20 0.41
SRC P12931 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042250 0.89 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DGAA
SCHEMBL13849020 0.83 PDE4A (0.79) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL13849014 0.76 PDE4A (0.65) PDE4APDE4BPDE4CPDE4D
SCHEMBL7434132 0.76 PDE4A (0.79) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL5846742 0.75 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DGAA
SCHEMBL13849056 0.74 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DCFD
SCHEMBL4037982 0.71 PDE4A (0.82) PDE4APDE4BPDE4CPDE4D
SCHEMBL4044216 0.71 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL4041704 0.70 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DCFD
SCHEMBL7435677 0.69 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487797-B1 HETERO-BRIDGE SUBSTITUTED 8-ARYLQUINOLINE PDE4 INHIBITORS MERCK FROSST CANADA LTD (CA) 2009-05-27 EP disclosed