SCHEMBL13849080

SCHEMBL13849080

CCS(=O)(=O)C(C)(C)c1cc(-c2cccc(CSc3ccccc3C(=O)OC)c2)c2ncccc2c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 15/20 0.51
PDE4A P27815 14/20 0.48
PDE4B Q07343 14/20 0.48
PDE4C Q08493 14/20 0.48
PDE4D Q08499 14/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039602 0.93 CYP2C9 (0.60) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4040252 0.79 CYP2C9 (0.56) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4039005 0.78 CYP2C9 (0.61) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4042502 0.77 CYP2C9 (0.60) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL13848926 0.76 PDE4A (0.56) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4041940 0.76 CYP2C9 (0.66) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4039163 0.75 CYP2C9 (0.67) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4039081 0.74 CYP2C9 (0.73) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4047138 0.72 CYP2C9 (0.62) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL4038639 0.72 PDE4A (0.78) CYP2C9PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487797-B1 HETERO-BRIDGE SUBSTITUTED 8-ARYLQUINOLINE PDE4 INHIBITORS MERCK FROSST CANADA LTD (CA) 2009-05-27 EP disclosed