SCHEMBL13858932

SCHEMBL13858932

C[C@]1(c2cc(Br)c(F)cc2F)OC(N)=NCC1(F)F

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.36
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1980420 0.80 BACE1 (0.41) BACE1CYP2D6
SCHEMBL13859218 0.78 BACE1 (0.49) BACE1CYP2D6
SCHEMBL1984301 0.77 CYP2D6 (0.33) CYP2D6
SCHEMBL13268451 0.74 BACE1 (0.38) BACE1
SCHEMBL13859156 0.74 BACE1 (0.45) BACE1
SCHEMBL13268504 0.74 BACE1 (0.32) BACE1CYP2D6
SCHEMBL14165303 0.74 BACE2 (0.44) BACE1
SCHEMBL1979221 0.74 BACE2 (0.44) BACE1
SCHEMBL13859149 0.73 MAPK1 (0.33)
SCHEMBL13859030 0.72 SMN1; SMN2 (0.33) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2709992-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. Hoffmann-La Roche AG (CH) 2014-03-26 EP disclosed
WO-2012156284-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2012-11-22 WO disclosed