SCHEMBL13858993

SCHEMBL13858993

C[C@]1(c2cc(NC3COC3)ccc2F)OC(N)=NCC1(F)F

nearest known ligand 0.48

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.48
BACE2 Q9Y5Z0 18/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13859466 0.92 BACE1 (0.59) BACE1BACE2
SCHEMBL1979443 0.81 BACE1 (0.51) BACE1BACE2
SCHEMBL13859237 0.80 BACE1 (0.55) BACE1BACE2
SCHEMBL13858956 0.79 BACE1 (0.48) BACE1BACE2
SCHEMBL13859504 0.79 BACE1 (0.41) BACE1BACE2
SCHEMBL1980420 0.79 BACE1 (0.41) BACE1BACE2
SCHEMBL1982738 0.77 BACE1 (0.61) BACE1BACE2
SCHEMBL1980997 0.77 BACE1 (0.42) BACE1BACE2
SCHEMBL13836168 0.76 BACE1 (0.57) BACE1BACE2
SCHEMBL13836169 0.76 BACE1 (0.57) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2709992-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. Hoffmann-La Roche AG (CH) 2014-03-26 EP claimed
WO-2012156284-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2012-11-22 WO claimed
EP-2709992-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. Hoffmann-La Roche AG (CH) 2014-03-26 EP disclosed
WO-2012156284-A1 1,3-OXAZINES AS BACE1 AND/OR BACE2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2012-11-22 WO disclosed