SCHEMBL1386083

SCHEMBL1386083

CC(CN)C1CN(c2c(F)cc3c(=O)n(N)c(=O)n(C4CC4)c3c2Cl)CC1(F)F

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CACNA1C Q13936 1/20 0.41
SCN5A Q14524 1/20 0.41
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1385392 0.90 KCNH2 (0.46) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4516872 0.86 KCNH2 (0.38) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4524309 0.81 KCNH2 (0.39) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4500385 0.80 KCNH2 (0.44) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6363485 0.79 KCNH2 (0.42) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4519134 0.78 KCNH2 (0.42) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1384915 0.78 KCNH2 (0.30) KCNH2
SCHEMBL4520780 0.78 KCNH2 (0.40) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1383915 0.77 KCNH2 (0.39) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1383918 0.77 KCNH2 (0.39) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4811978-B2 2011-11-09 JP claimed
EP-1255739-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2002-11-13 EP claimed
WO-2001053273-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2001-07-26 WO claimed