SCHEMBL13861995

SCHEMBL13861995

C=C/N=C\N(C)c1ccc2nc(NC(=O)c3ccc(C(C)(C)C)cc3)cn2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 13/20 0.50
RET P07949 2/20 0.43
CDK2 P24941 2/20 0.43
GSK3B P49841 2/20 0.43
ITK Q08881 2/20 0.43
MERTK Q12866 2/20 0.43
PRKAA1 Q13131 2/20 0.43
ROCK1 Q13464 2/20 0.43
MAP3K6 O95382 2/20 0.42
CSNK1D P48730 3/20 0.40
CSNK1E P49674 3/20 0.40
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
CHRM1 P11229 1/20 0.39
DRD2 P14416 1/20 0.39
ADRA2B P18089 1/20 0.39
DRD1 P21728 1/20 0.39
HRH2 P25021 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR1D P28221 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13498801 0.87 MAP3K5 (0.59) MAP3K5RETCDK2GSK3BITK
Hydrochloric Acid SCHEMBL3485897 0.86 MAP3K5 (0.58) MAP3K5RETCDK2GSK3BITK
SCHEMBL13498928 0.77 MAP3K5 (0.53) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486150 0.77 MAP3K5 (0.66) MAP3K5RETCDK2GSK3BITK
SCHEMBL13498941 0.77 MAP3K5 (0.53) MAP3K5RETCDK2GSK3BITK
SCHEMBL3485708 0.76 MAP3K5 (0.61) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486218 0.76 MAP3K5 (0.61) MAP3K5RETCDK2GSK3BITK
SCHEMBL3485883 0.76 MAP3K5 (0.65) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486292 0.75 MAP3K5 (0.60) MAP3K5RETCDK2GSK3BITK
Hydrochloric Acid SCHEMBL3486257 0.75 MAP3K5 (0.60) MAP3K5RETCDK2GSK3BITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058309-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-05-13 EP disclosed